Highly efficient methods for the one-pot synthesis of beta-substituted enones.
نویسندگان
چکیده
A mild and practically-convenient one-pot procedure for the direct beta-substitution of enones has been developed using a conjugate addition-oxidation strategy with a full range of copper-based reagents and N-tert-butylphenylsulfinimidoyl chloride; alkyl- and aryl-substituted enones are delivered in good to excellent yields.
منابع مشابه
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ورودعنوان ژورنال:
- Organic & biomolecular chemistry
دوره 4 1 شماره
صفحات -
تاریخ انتشار 2006